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ANTIVIRAL WHO Essential Verified Rx Required
Valacyclovir
Also known as:Valtrex "Valtrex"
2 Protocols
2 views
Primary Use
Treatment and suppression of herpes infections.
Also Used For:
Shingles
Cold sores
Herpes suppression
Drug Classification
Medication Type
ANTIVIRAL
Drug Class
Nucleoside analogue prodrug
Dosage & Administration
Standard Dosage
500mg-1g
Frequency
Once or twice daily
Duration
3-10 days for outbreaks, long-term for suppression
Route
ORAL
Best Time
Same time each day
Important
Full glass of water
Available Forms
Dosage Forms
TABLETCAPSULE
Available Strengths
500mg1g
Appearance
Blue caplet
Effectiveness
Success Rate
Similar to acyclovir with better bioavailability
Cross-resistance with acyclovir. Rare in immunocompetent individuals.
Treatment Protocols
Herpes - Daily Suppressive Therapy
For: HERPES_SIMPLEX
Dosage
500mg
Frequency
Once daily
Duration
Ongoing (typically 1 year minimum)
Reduces outbreaks by 70-80%. Reduces transmission by ~50%.
Herpes - Episodic Treatment
For: HERPES_SIMPLEX
Dosage
1g (1000mg)
Frequency
Twice daily
Duration
1 day
Reduces outbreak duration by 1-2 days
Safety Information
Common Side Effects
HeadacheNauseaAbdominal painDizziness
Serious Side Effects (Seek Medical Help)
Kidney problems
Neurological effects
Blood disorders
Contraindications (Do Not Use If)
Valacyclovir allergy
Severe kidney impairment
Drug Interactions
Other nephrotoxic drugsCimetidineProbenecid
Pregnancy
Category B - Generally safe
Breastfeeding
Compatible with breastfeeding
Pricing Information
Mfg. Cost
$3
Global Avg. Price
$25
Patent Status
Brand and generic available
Prices may vary significantly by country, pharmacy, and insurance coverage. This is an average estimate.
Availability & Regulations
Prescription Required
Not OTC
Not Controlled
FDA Approval
1995
Available In
π΅πPhilippinesπΉπThailandπ»π³VietnamπΈπ¬Singaporeπ²πΎMalaysiaπΊπΈUnited Statesπ¬π§United Kingdom